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作者(2019)在《Synthesis and insecticidal bioactivities of 2,3-dihydroimidazo[1,2-a] pyridin-5(1H)-one derivatives》一文中研究指出:A novel synthesis of 2,3-dihydroimidazo[1,2-a]pyridin-5 (1H)-one 4 and its derivatives were described.Preliminary bioassays showed that some of the target compounds exhibited excellent insecticidal activities against brown planthopper (Nilaparvata lugens), cowpea aphids (Aphis craccivora) (4,5 a, 5 c, 5 g,5 h, 5 j, 5 r, 6 b, 6 e) and carmine spider mite (Tetranychus cinnabarinus (5 f, 5 s, 6 a) at 500 mg/L. Among them,compound 4 was still active against brown planthopper and cowpea aphids at 4 mg/L. The insecticidal activities were influenced by the types and position of the substituents, which provided guidance for the structure modifications.
Abstract
A novel synthesis of 2,3-dihydroimidazo[1,2-a]pyridin-5 (1H)-one 4 and its derivatives were described.Preliminary bioassays showed that some of the target compounds exhibited excellent insecticidal activities against brown planthopper (Nilaparvata lugens), cowpea aphids (Aphis craccivora) (4,5 a, 5 c, 5 g,5 h, 5 j, 5 r, 6 b, 6 e) and carmine spider mite (Tetranychus cinnabarinus (5 f, 5 s, 6 a) at 500 mg/L. Among them,compound 4 was still active against brown planthopper and cowpea aphids at 4 mg/L. The insecticidal activities were influenced by the types and position of the substituents, which provided guidance for the structure modifications.
论文参考文献
[1].Synthesis and insecticidal evaluation of tetrahydroimidazo[1,2-a]pyridin-5(1H)-one derivatives[J]. Xuan-Qi Liu,Ya-Qin Liu,Xu-Sheng Shao,Zhi-Ping Xu,Xiao-Yong Xu,Zhong Li.  Chinese Chemical Letters.2016(01)[2].Semisynthesis of new ethers from furyl-ring-based acylation derivatives of fraxinellone as insecticidal agents against Mythimna separata Walker in vivo[J]. Ruige Yang,Yong Guo,Yuanyuan Zhang,Hui Xu.  Chinese Chemical Letters.2018(06)[3].Design,synthesis and insecticidal activities of novel anthranilic diamides containing fluorinated groups as potential ryanodine receptors activitors[J]. Chang-Chun Wu,Bao-Lei Wang,Jing-Bo Liu,Wei Wei,Yu-Xin Li,Yang Liu,Ming-Gui Chen,Li-Xia Xiong,Na Yang,Zheng-Ming Li.  Chinese Chemical Letters.2017(06)[4].Synthesis and insecticidal evaluation of phytoalexin phenalenones derivatives[J]. Ya-Nan Zhang,Yi-An Feng,Zhong Li,Xu-Sheng Shao.  Chinese Chemical Letters.2017(06)[5].Synthesis and insecticidal activities of 1,8-naphthyridine derivatives[J]. Qing-Qing Hou,Yi-Fei Jing,Xu-Sheng Shao.  Chinese Chemical Letters.2017(08)[6].Synthesis,insecticidal and acaricidal activities of novel 2-arylpyrroles[J]. LIU AiPing,TANG Ming,YU ShuYing,LIU XingPing,WANG XiaoGuang,PEI Hui,WU DaoXin,HU Li,OU XiaoMing,HUANG MingZhi.  Science China(Chemistry).2013(01)[7].Synthesis and insecticidal activities of novel bridged-neonicotinoids[J]. Dong-Dong Zhang,Shu-Xia Cui,Zhi-Ping Xu,Dong-Mei Li,Zhong-Zhen Tian.  Chinese Chemical Letters.2017(08)[8].Facile three-component synthesis and insecticidal evaluation of hexahydroimidazo[1,2-a]pyridine derivatives[J]. Ye-Feng Fan,Wen-Wen Zhang,Xu-Sheng Shao,Zhi-Ping Xu,Xiao-Yong Xu,Zhong Li.  Chinese Chemical Letters.2015(01)[9].Synthesis and insecticidal activities of new pyrethroid acid oxime ester derivatives[J]. MA Jun’an, HUANG Runqiu and CHAI Youxin(Institute and State Key Laboratory of Elemento-organic Chemistry, Nankai University, Tianjin 300071, China).  Progress in Natural Science.2002(04)[10].Study on the insecticidal activities of the extracts from four plants under orthogonal test[J]. WEN Pu-hong,ZHAO Wei-xing,WANG Yan,ZHAO Yong-chun,LI Zong-xiao(Key Laboratory for Phytochemistry of Shaanxi Province,Dept.Chem.& Chem.Eng.,Baoji University of Arts and Sciences,Baoji 721013,Shaanxi,China).  宝鸡文理学院学报(自然科学版).2012(01)
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:Synthesis and insecticidal bioactivities of 2,3-dihydroimidazo[1,2-a] pyridin-5(1H)-one derivatives论文
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